SCHEMBL7967329

SCHEMBL7967329

Cc1cc(C)cc(-c2c([C@H](C)COCc3ccccc3)c3cc(C(C)(C)C(=O)N4C5CCC4CC5)cnc3n2C(=O)OC(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.43
GNRHR P30968 18/20 0.39
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967331 1.00 CACNA1B (0.43) CACNA1BGNRHRCYP3A4
SCHEMBL8479412 0.92 GNRHR (0.44) GNRHRCYP3A4
SCHEMBL8479408 0.92 GNRHR (0.44) GNRHRCYP3A4
SCHEMBL7980867 0.87 CACNA1B (0.46) CACNA1BGNRHRCYP3A4
SCHEMBL7980869 0.87 CACNA1B (0.46) CACNA1BGNRHRCYP3A4
SCHEMBL8183827 0.87 CACNA1B (0.54) CACNA1BGNRHRCYP3A4
SCHEMBL8183825 0.87 CACNA1B (0.54) CACNA1BGNRHRCYP3A4
SCHEMBL8023243 0.86 CACNA1B (0.43) CACNA1BGNRHR
SCHEMBL8023239 0.86 CACNA1B (0.43) CACNA1BGNRHR
SCHEMBL7977562 0.80 GNRHR (0.51) CACNA1BGNRHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228867-B1 2-PHENYL-PYRROLO(2,3-B)PYRIDINE DERIVATIVES FOR TREATING UROGENITAL AND SLEEP DISORDERS; ANTICARCINOGENIC AGENTS; BENIGN PROSTATIC HYPERPLASIA MERCK & CO., INC. 2001-05-08 US disclosed
US-6110931-A FOR PREGNANCY PROPHYLAXIS AND TREATMENT OF GLANDULAR DISORDERS, HORMONE DEFICIENCY DISORDERS, GASTROINTESTINAL DISORDERS, GROWTH DISORDERS MERCK & CO., INC. (US) 2000-08-29 US disclosed