SCHEMBL7969276

SCHEMBL7969276

C=Cc1ccc(Cl)nc1NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LCK P06239 6/20 0.40
ATR Q13535 1/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40
ADORA3 P0DMS8 1/20 0.37
ADORA2B P29275 1/20 0.37
BRD4 O60885 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OGFRL1 Q5TC84 1/20 0.37
MAPKAPK2 P49137 2/20 0.37
LMNA P02545 1/20 0.37
ACSS2 Q9NR19 1/20 0.36
SYK P43405 1/20 0.36
NAMPT P43490 1/20 0.36
MAP4K4 O95819 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29541653 0.87 ATR (0.44) LCKATRKMT2AMEN1NPC1
SCHEMBL4056822 0.87 ATR (0.44) LCKATRKMT2AMEN1NPC1
SCHEMBL10270535 0.84 LCK (0.39) LCKATRKMT2AMEN1NPC1
SCHEMBL30301479 0.78 ATR (0.43) LCKATRKMT2AMEN1NPC1
SCHEMBL10270285 0.77 ATR (0.45) LCKATRKMT2AMEN1NPC1
SCHEMBL4059749 0.76 ATR (0.41) LCKATRKMT2AMEN1NPC1
SCHEMBL1514112 0.76 ATR (0.56) LCKATRKMT2ANPC1RAB9A
SCHEMBL4053414 0.75 ATR (0.40) LCKATRKMT2AMEN1NPC1
SCHEMBL21605114 0.75 MAPKAPK2 (0.41) LCKATRMAPKAPK2
SCHEMBL30629718 0.75 MAPKAPK2 (0.41) LCKATRMAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010012398-A1 SUBSTITUTED PYRIDINES, AND USE THEREOF AS GSK3 INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-04 WO disclosed
WO-2009138176-A1 SUBSTITUTED IMIDAZO- AND TRIAZOLOPYRIMIDINES, IMIDAZO- AND PYRAZOLOPYRAZINES AND IMIDAZOTRIAZINES AS GSK3BETA-INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-11-19 WO disclosed
WO-2009074259-A1 TRIAZOLOTRIAZINES AND TRIAZOLOPYRAZINES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-06-18 WO disclosed
WO-2009007029-A1 IMIDAZO-, PYRAZOLOPYRAZINES AND IMIDAZOTRIAZINES AND THEIR USE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-01-15 WO disclosed
WO-2008113469-A2 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-09-25 WO disclosed