SCHEMBL7970075

SCHEMBL7970075

Cc1ccc(N)c(-n2ccnc2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.66
MAPT P10636 3/20 0.44
LMNA P02545 2/20 0.44
CYP19A1 P11511 3/20 0.42
CYP11B1 P15538 3/20 0.42
CYP11B2 P19099 3/20 0.42
CYP3A4 P08684 4/20 0.41
TDP1 Q9NUW8 2/20 0.41
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
ALOX15 P16050 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL997561 0.86 IDO1 (0.53) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL11569176 0.82 IDO1 (0.44) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL13242920 0.79 IDO1 (0.66) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL2666052 0.79 CYP19A1 (0.45) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL25822705 0.79 IDO1 (0.66) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL11705217 0.79 IDO1 (0.66) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL1885632 0.79 CYP3A4 (0.46) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL14121087 0.77 CYP11B1 (0.61) MAPTLMNACYP19A1CYP11B1CYP11B2
SCHEMBL11846584 0.77 IDO1 (0.43) IDO1MAPTLMNACYP19A1CYP11B1
SCHEMBL16559778 0.77 CYP2D6 (0.44) IDO1MAPTLMNACYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO disclosed