SCHEMBL7970206

SCHEMBL7970206

CCc1nc(Oc2ccc(CC(C)(C)NC[C@H](O)COc3cccc4[nH]ccc34)cc2)ccc1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 17/20 0.53
ADRB1 P08588 5/20 0.52
ADRB2 P07550 5/20 0.52
CYP2D6 P10635 2/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A4 P31645 1/20 0.49
CASR P41180 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KCNH2 Q12809 1/20 0.49
KDM4E B2RXH2 1/20 0.46
USP2 O75604 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
THRB P10828 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7970203 1.00 ADRB3 (0.53) ADRB3ADRB1ADRB2CYP2D6SLC6A2
SCHEMBL7973558 0.91 ADRB3 (0.54) ADRB3ADRB1ADRB2CYP2D6SLC6A2
SCHEMBL7973555 0.91 ADRB3 (0.54) ADRB3ADRB1ADRB2CYP2D6SLC6A2
SCHEMBL7973641 0.87 ADRB3 (0.67) ADRB3ADRB1ADRB2
SCHEMBL7976392 0.87 ADRB3 (0.67) ADRB3ADRB1ADRB2
SCHEMBL6387352 0.84 ADRB3 (0.51) ADRB3ADRB1ADRB2CYP2D6SLC6A2
SCHEMBL6387355 0.84 ADRB3 (0.51) ADRB3ADRB1ADRB2CYP2D6SLC6A2
SCHEMBL7746703 0.82 ADRB3 (0.49) ADRB3ADRB1ADRB2CYP2D6SLC6A2
SCHEMBL7746708 0.82 ADRB3 (0.49) ADRB3ADRB1ADRB2CYP2D6SLC6A2
SCHEMBL7970016 0.81 ADRB3 (0.77) ADRB3ADRB1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001036412-A1 PROCESS FOR THE PREPARATION OF ARYLOXY PROPANOLAMINES ELI LILLY AND COMPANY (US) 2001-05-25 WO disclosed