SCHEMBL7970762

SCHEMBL7970762

COc1c(-c2ccccc2)nn(C)c1-c1nc2cc(F)c(C)cc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 4/20 0.44
KDM4E B2RXH2 5/20 0.42
HSD17B10 Q99714 4/20 0.42
TP53 P04637 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
MAPT P10636 4/20 0.39
KMT2A Q03164 2/20 0.39
GAPDH P04406 1/20 0.39
GUSB P08236 2/20 0.39
ADORA3 P0DMS8 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10140093 0.87 TP53 (0.38) AMY1AKDM4EHSD17B10TP53ALDH1A1
SCHEMBL10172619 0.87 DHODH (0.39) AMY1AKDM4EHSD17B10TP53ALDH1A1
SCHEMBL10140097 0.85 DHODH (0.41) KDM4EHSD17B10TP53ALDH1A1HPGD
SCHEMBL7982191 0.83 P2RY6 (0.51) KDM4EHSD17B10TP53ALDH1A1HPGD
SCHEMBL10139799 0.82 NPC1 (0.65) KDM4EHSD17B10TP53ALDH1A1HPGD
SCHEMBL7959879 0.81 KDM4E (0.40) AMY1AKDM4EHSD17B10TP53ALDH1A1
SCHEMBL7961586 0.79 CHEK2 (0.53) KDM4EALDH1A1HPGDSMN1; SMN2NPC1
SCHEMBL7966178 0.78 NPC1 (0.65) KDM4EHSD17B10TP53ALDH1A1HPGD
SCHEMBL10140405 0.78 CHEK2 (0.48) KDM4EHSD17B10TP53ALDH1A1HPGD
SCHEMBL7960793 0.77 KDM4E (0.52) KDM4EHSD17B10TP53ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed