SCHEMBL7972482

SCHEMBL7972482

CC(=O)N1CCN(NC(=O)c2ccc(N(C)C)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.49
HDAC1 Q13547 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
ITK Q08881 11/20 0.46
ALDH1A1 P00352 2/20 0.45
POLB P06746 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
NAMPT P43490 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972839 0.83 CYP2D6 (0.53) CYP2D6HDAC6ALDH1A1MAPTHPGD
SCHEMBL8018069 0.83 CYP2D6 (0.53) CYP2D6HDAC6ALDH1A1MAPTHPGD
SCHEMBL7972620 0.82 CYP2D6 (0.60) CYP2D6ALDH1A1POLB
SCHEMBL194951 0.82 CYP2D6 (0.72) CYP2D6ALDH1A1MAPTHPGDHTT
SCHEMBL14590778 0.81 HTT (0.65) CYP2D6HDAC6MAPTHTT
SCHEMBL7968909 0.81 CYP2D6 (0.50) CYP2D6ALDH1A1TDP1MAPTHPGD
Water SCHEMBL3089403 0.81 CYP2D6 (0.70) CYP2D6ALDH1A1MAPTHPGDHTT
SCHEMBL7972123 0.79 CYP2D6 (0.52) CYP2D6MAPTHPGDHTT
SCHEMBL7975155 0.79 HPGD (0.50) CYP2D6HDAC1HDAC6ALDH1A1MAPT
SCHEMBL7970177 0.79 PLK1 (0.50) CYP2D6ALDH1A1POLBMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291464-B1 POTENTIATION OF THE CHOLINERGIC ACTIVITY; THERAPEUTIC TREATMENT OF AMNESIA, DEMENTIA OR SENILE DEMENTIA FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-09-18 US disclosed
EP-0968201-A2 NEW AMINOPIPERAZINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-01-05 EP disclosed
WO-1998035951-A2 NEW AMINOPIPERAZINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-08-20 WO disclosed