SCHEMBL7974049

SCHEMBL7974049

CCOC(=O)C=Cc1ccc2c(c1)CN(C(=O)O)CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.51
DPP4 P27487 1/20 0.51
HPGD P15428 3/20 0.51
MAPT P10636 2/20 0.51
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 1/20 0.51
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
MAOB P27338 3/20 0.47
CYP3A4 P08684 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46
FDPS P14324 1/20 0.46
HTR1A P08908 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974045 1.00 TTR (0.51) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL20995788 0.95 TTR (0.51) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL20995789 0.95 TTR (0.51) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL20509948 0.93 TTR (0.53) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL20509947 0.93 TTR (0.53) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL20509713 0.89 TTR (0.49) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL20509714 0.89 TTR (0.49) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL27766220 0.87 KDM4E (0.48) TTRHPGDMAPTALDH1A1KDM4E
SCHEMBL8194148 0.87 TTR (0.54) TTRDPP4HPGDMAPTALDH1A1
SCHEMBL8194154 0.87 TTR (0.54) TTRDPP4HPGDMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200978-B1 FOR PREVENTING OR TREATING INFLAMMATORY DISEASES SUCH AS ARTHRITIS, PSORIASIS, ASTHMA, OR INFLAMMATORY BOWEL DISEASE, DISORDERS OF RESPIRATORY FUNCTION, GASTROINTESTINAL DISORDERS SUCH AS FUNCTIONAL BOWEL DISEASE, AS ANALGESICS PFIZER INC. 2001-03-13 US disclosed
WO-2000007993-A1 SUBSTITUTED ISOQUINOLEINES AND THEIR USE AS ANTICONVULSIVANTS SMITHKLINE BEECHAM PLC (GB) 2000-02-17 WO disclosed