SCHEMBL7975422

SCHEMBL7975422

FC(F)(F)c1cc(CNCC(c2ccccc2)N2CCN(CCc3ccc(Cl)cc3)CC2)cc(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 7/20 0.55
TACR1 P25103 11/20 0.50
CCR2 P41597 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7932641 0.93 CCR3 (0.57) CCR3TACR1CCR2
SCHEMBL7925814 0.91 CCR3 (0.50) CCR3TACR1CYP2D6
SCHEMBL7938489 0.88 CCR3 (0.59) CCR3TACR1CYP2D6
SCHEMBL16226687 0.85 TACR1 (0.52) CCR3TACR1
SCHEMBL7987228 0.82 CCR3 (0.67) CCR3TACR1CCR2
SCHEMBL7938403 0.82 CCR3 (0.59) CCR3TACR1CYP2D6
SCHEMBL7926034 0.80 TACR1 (0.48) CCR3TACR1
SCHEMBL7934653 0.79 CCR3 (0.60) CCR3TACR1
SCHEMBL6479126 0.79 TACR1 (0.54) CCR3TACR1CCR2
SCHEMBL8674953 0.78 TACR1 (0.45) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191135-B1 Neurokinin antagonists BOEHRINGER INGELHEIM KG (DE) 2001-02-20 US claimed
US-6191135-B1 Neurokinin antagonists BOEHRINGER INGELHEIM KG (DE) 2001-02-20 US disclosed
WO-1996008480-A1 NEUROKININ ANTAGONISTS BOEHRINGER INGELHEIM KG (DE) 1996-03-21 WO disclosed