SCHEMBL7978153

SCHEMBL7978153

Cc1nc2ccccn2c1-c1ccnc(Nc2ccc(C(=O)NOC3CCCCO3)cc2F)n1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.51
CDK2 P24941 6/20 0.49
CCNE1 P24864 4/20 0.49
CDK4 P11802 4/20 0.49
INSR P06213 4/20 0.46
IGF1R P08069 6/20 0.46
EGFR P00533 3/20 0.46
ERBB2 P04626 3/20 0.46
MAPK14 Q16539 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980583 0.86 CDK2 (0.50) HDAC1CDK2CCNE1CDK4
SCHEMBL10252325 0.86 CDK2 (0.49) HDAC1CDK2CCNE1CDK4INSR
SCHEMBL10252165 0.85 CDK2 (0.49) HDAC1CDK2CCNE1CDK4INSR
SCHEMBL10252196 0.83 CDK2 (0.51) HDAC1CDK2CCNE1CDK4
SCHEMBL10252153 0.82 CDK2 (0.50) HDAC1CDK2CCNE1CDK4INSR
SCHEMBL7978154 0.82 CDK2 (0.50) HDAC1CDK2CCNE1CDK4INSR
SCHEMBL7964023 0.82 CDK2 (0.50) HDAC1CDK2CCNE1CDK4
SCHEMBL699844 0.82 HDAC1 (0.59) HDAC1CDK2CCNE1CDK4INSR
SCHEMBL7978108 0.82 CDK2 (0.62) HDAC1CDK2CCNE1CDK4INSR
SCHEMBL7965090 0.82 CDK2 (0.49) HDAC1CDK2CCNE1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010009155-A2 FUSED HETEROCYCLYC INHIBITOR COMPOUNDS GILEAD COLORADO, INC. (US) 2010-01-21 WO disclosed