SCHEMBL7980648

SCHEMBL7980648

N#Cc1ccc(C(c2ccc(Cl)cc2)n2ccnc2)cc1F

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 16/20 0.63
CYP1A2 P05177 3/20 0.51
CYP3A4 P08684 3/20 0.51
CYP2D6 P10635 3/20 0.51
FNTA P49354 1/20 0.45
FNTB P49356 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507798 0.80 CYP19A1 (0.85) CYP19A1CYP1A2CYP3A4CYP2D6
SCHEMBL10693298 0.80 CYP19A1 (1.00) CYP19A1CYP1A2CYP3A4CYP2D6
SCHEMBL3499887 0.77 FNTA (0.59) CYP19A1CYP1A2CYP3A4CYP2D6FNTA
SCHEMBL11366789 0.74 CYP19A1 (1.00) CYP19A1CYP1A2CYP3A4CYP2D6FNTA
SCHEMBL8917184 0.73 CYP19A1 (0.84) CYP19A1CYP1A2CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL7980448 0.73 FNTA (0.51) CYP19A1FNTAFNTB
SCHEMBL1507825 0.72 CYP19A1 (1.00) CYP19A1CYP3A4
SCHEMBL11479567 0.71 CYP19A1 (0.68) CYP19A1CYP1A2CYP3A4CYP2D6FNTA
SCHEMBL11463766 0.71 CYP19A1 (0.68) CYP19A1CYP1A2CYP3A4CYP2D6FNTA
SCHEMBL11353276 0.71 CYP19A1 (0.91) CYP19A1CYP1A2CYP3A4CYP2D6FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6297239-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2001-10-02 US disclosed