SCHEMBL7983262

SCHEMBL7983262

CC(C)(C)c1ccc2c(c1)nc(Nc1ccccc1Br)c1c(P(=O)(O)O)ncn12

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LCK P06239 6/20 0.41
RAF1 P04049 2/20 0.36
BRAF P15056 1/20 0.36
TP53 P04637 2/20 0.35
EGFR P00533 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.31
POLB P06746 1/20 0.31
NPC1 O15118 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981071 0.92 LCK (0.41) LCKRAF1BRAFTP53EGFR
SCHEMBL7970045 0.90 LCK (0.53) LCKTP53ALDH1A1MAPTPOLB
SCHEMBL7970141 0.86 LCK (0.56) LCKTP53ALDH1A1MAPTABCG2
SCHEMBL7981479 0.84 LCK (0.35) LCKALDH1A1MAPTPOLBNPC1
SCHEMBL7969544 0.83 LCK (0.40) LCK
SCHEMBL7983573 0.83 LCK (0.43) LCKRAF1BRAFTP53ALDH1A1
SCHEMBL7969561 0.82 LCK (0.41) LCKTP53MAPT
SCHEMBL7979971 0.78 LCK (0.69) LCK
SCHEMBL7969727 0.74 LCK (0.67) LCKTP53ALDH1A1MAPTNPC1
SCHEMBL7979942 0.71 LCK (0.56) LCKTP53MAPTPOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed