SCHEMBL7984411

SCHEMBL7984411

CC(Nc1nccc(-n2cnc3ccncc32)n1)C1CCCN(C(=O)OCc2ccccc2)C1

nearest known ligand 0.88

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LCK P06239 18/20 0.88
IDH1 O75874 1/20 0.52
JAK2 O60674 1/20 0.51
JAK3 P52333 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984542 0.93 LCK (1.00) LCKIDH1
SCHEMBL7586925 0.89 LCK (0.81) LCKIDH1
SCHEMBL7552112 0.86 LCK (0.80) LCKIDH1
SCHEMBL7549251 0.84 LCK (0.78) LCKIDH1
SCHEMBL7986922 0.84 LCK (0.83) LCK
SCHEMBL7506710 0.83 LCK (0.74) LCKJAK2JAK3
SCHEMBL7547222 0.83 LCK (0.76) LCKIDH1
SCHEMBL7504117 0.82 LCK (1.00) LCK
SCHEMBL7972879 0.82 LCK (1.00) LCK
SCHEMBL7542450 0.81 LCK (0.77) LCKIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329380-B1 PYRIMIDINE BENZIMIDIZAZOLE, PYRIMIDINEIMIDAZOLE OR PYRIDINE IMIDAZOLE COMPOUNDS FOR ANTICANCER AGENTS OR ATHEROSCLEROSIS MERCK & CO., INC. 2001-12-11 US disclosed