SCHEMBL7984478

SCHEMBL7984478

CCOC(=O)[C@@H]1C[C@H]2C[C@@H](COCC#N)CC[C@H]2CN1C(=O)OC

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.33
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
CYP3A4 P08684 2/20 0.31
KDM4E B2RXH2 1/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6605879 1.00 IDH1 (0.33) IDH1HCRTR1HCRTR2CYP3A4KDM4E
SCHEMBL6605662 0.85 JAK1 (0.35) IDH1HCRTR1HCRTR2CYP3A4KDM4E
SCHEMBL8440718 0.84 IDH1 (0.37) IDH1KDM4EDPP4
SCHEMBL6606285 0.84 IDH1 (0.33) IDH1CYP3A4KDM4EDPP4DPP8
SCHEMBL6605287 0.83 IDH1 (0.33) IDH1CYP3A4KDM4EDPP4DPP8
SCHEMBL6791730 0.82 NR1H2 (0.36) CYP3A4KDM4E
SCHEMBL6328305 0.82 NR1H2 (0.36) CYP3A4KDM4E
SCHEMBL6324214 0.82 CYP3A4 (0.34) CYP3A4KDM4E
SCHEMBL6605366 0.81 CYP3A4 (0.34) CYP3A4KDM4E
SCHEMBL6608201 0.81 CYP3A4 (0.34) CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242462-B1 NOVEL DECAHYDROISOQUINOLINE DERIVATIVES WHICH ARE SELECTIVE GLUR5 RECEPTOR ANTAGONISTS. ELI LILLY AND COMPANY 2001-06-05 US disclosed