SCHEMBL7986683

SCHEMBL7986683

OCCCCCCNCc1ccccc1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 1/20 0.56
CA12 O43570 4/20 0.51
CA2 P00918 4/20 0.51
CA9 Q16790 4/20 0.51
CHRM2 P08172 6/20 0.47
KDM4E B2RXH2 2/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GRIN1 Q05586 3/20 0.43
GRIN2A Q12879 3/20 0.43
BCHE P06276 2/20 0.43
ACHE P22303 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16466899 0.87 SCN8A (0.54) SCN8ACA12CA2CA9KDM4E
SCHEMBL25590510 0.84 SCN8A (0.59) SCN8ACA12CA2CA9CHRM2
SCHEMBL7077084 0.83 SCN8A (0.60) SCN8ACA12CA2CA9CHRM2
SCHEMBL13975078 0.81 SCN8A (0.62) SCN8ACA12CA2CA9CHRM2
SCHEMBL13436118 0.79 SCN8A (0.54) SCN8AKDM4ETSHRALDH1A1HTT
SCHEMBL17274380 0.78 HDAC1 (0.52) KDM4EALDH1A1
SCHEMBL21674183 0.77 SCN8A (0.57) SCN8AKDM4EALDH1A1HTTTDP1
SCHEMBL16269037 0.77 SCN8A (0.54) SCN8ACA12CA2KDM4EALDH1A1
SCHEMBL10925708 0.76 CHRM2 (0.80) CA12CA2CA9CHRM2TSHR
SCHEMBL17400756 0.76 CA12 (0.56) CA12CA2CA9CHRM2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6214833-B1 MADE BY ACYLATION ZAMBON GROUP S.P.A. (IT) 2001-04-10 US disclosed
EP-0970075-A1 PYRIMIDINONE-1,3-OXATHIOLANE DERIVATIVES WITH ANTIVIRAL ACTIVITY ZAMBON GROUP S.p.A. (IT) 2000-01-12 EP disclosed
WO-1998043972-A1 PYRIMIDINONE-1,3-OXATHIOLANE DERIVATIVES WITH ANTIVIRAL ACTIVITY ZAMBON GROUP S.P.A. (IT) 1998-10-08 WO disclosed