SCHEMBL7986793

SCHEMBL7986793

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SCCc3cn4cccnc4n3)[C@H](C)[C@H]12

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.38
ESR1 P03372 1/20 0.38
PTGS1 P23219 1/20 0.38
PDE4A P27815 1/20 0.38
ALDH1A1 P00352 8/20 0.36
KDM4E B2RXH2 7/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 5/20 0.36
HSD17B10 Q99714 3/20 0.36
NPC1 O15118 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RCE1 Q9Y256 1/20 0.34
RECQL P46063 1/20 0.34
RAB9A P51151 1/20 0.34
PDE10A Q9Y233 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ABCC2 Q92887 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987037 1.00 CACNA1C (0.38) CACNA1CESR1PTGS1PDE4AALDH1A1
SCHEMBL7982633 0.85 PTGS1 (0.40) CACNA1CESR1PTGS1PDE4AALDH1A1
SCHEMBL7982891 0.85 PTGS1 (0.40) CACNA1CESR1PTGS1PDE4AALDH1A1
SCHEMBL7969463 0.83 CACNA1C (0.39) CACNA1CESR1PTGS1PDE4AKDM4E
SCHEMBL7987229 0.83 CACNA1C (0.38) CACNA1CESR1PTGS1PDE4AKDM4E
SCHEMBL7983336 0.83 CACNA1C (0.38) CACNA1CESR1PTGS1PDE4AKDM4E
SCHEMBL7980451 0.80 ESR1 (0.40) CACNA1CESR1PTGS1PDE4AKDM4E
SCHEMBL7969529 0.80 CACNA1C (0.40) CACNA1CESR1PTGS1PDE4AKDM4E
SCHEMBL7969417 0.80 CACNA1C (0.40) CACNA1CESR1PTGS1PDE4AKDM4E
SCHEMBL7979837 0.79 CACNA1C (0.41) CACNA1CESR1PTGS1PDE4AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed