SCHEMBL7986884

SCHEMBL7986884

CCOC(=O)CCCN1CCn2nc(C(=O)O)cc2C1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TNF P01375 10/20 0.37
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CHRM1 P11229 2/20 0.35
SLC6A2 P23975 1/20 0.35
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31607767 0.77 HDAC6 (0.36) ALDH1A1SIGMAR1CYP4F2CYP4A11
SCHEMBL6474034 0.77 POLB (0.50) TNFMAPTALDH1A1
SCHEMBL11861074 0.73 CYP1A2 (0.53) TNFGAAALDH1A1HSD17B10HRH2
SCHEMBL3310783 0.72 HDAC6 (0.41) ALDH1A1CYP4F2CYP4A11
SCHEMBL6474441 0.72 POLB (0.52) ALDH1A1
SCHEMBL3309074 0.71 CYP1A2 (0.40) GAAALDH1A1HSD17B10
SCHEMBL31389960 0.71 P2RY14 (0.35) CYP4F2CYP4A11
SCHEMBL31389811 0.71 MAPT (0.37) MAPT
SCHEMBL1127701 0.69 PAOX (0.51) TNFALDH1A1HRH2HRH1
SCHEMBL30887203 0.68 CYP1A2 (0.47) TNFGAAALDH1A1HRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207663-B1 AS INHIBITORS OF BONE RESORPTION, TUMOR GROWTH, TUMOR METASTASIS, OR INFLAMMATION, OR FOR THE TREATMENT OR PROPHYLAXIS OF CARDIOVASCULAR DISORDERS, NEPHROPATHIES OR RETINOPATHIES HOECHST ATKIENGESELLSCHAFT (DE) 2001-03-27 US disclosed