SCHEMBL7989695

SCHEMBL7989695

O=C1CC(C#CC2CC2)(C(F)(F)F)c2c(ccc(F)c2F)N1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 8/20 0.66
HTR2A P28223 2/20 0.42
NR1I2 O75469 1/20 0.42
NR3C1 P04150 1/20 0.42
PGR P06401 1/20 0.42
ADRB1 P08588 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
MAPT P10636 1/20 0.42
CNR1 P21554 1/20 0.42
SLC6A2 P23975 1/20 0.42
HTR2C P28335 1/20 0.42
MAPK1 P28482 1/20 0.42
AGTR1 P30556 1/20 0.42
CCKBR P32239 1/20 0.42
PPARG P37231 1/20 0.42
OPRK1 P41145 1/20 0.42
SLC6A3 Q01959 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE3A Q14432 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7975568 0.80 CYP46A1 (1.00) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL4576238 0.76 CYP46A1 (0.43) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL29400467 0.76 CYP46A1 (0.43) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL1152387 0.76 CYP46A1 (0.43) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL7473677 0.74 CYP46A1 (0.42) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL7808948 0.73 CYP46A1 (0.41) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL7910312 0.73 CYP46A1 (0.41) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL7811865 0.73 CYP46A1 (0.41) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL1151379 0.71 CYP46A1 (0.46) CYP46A1HTR2ANR1I2NR3C1PGR
SCHEMBL1152275 0.71 CYP46A1 (0.50) CYP46A1HTR2ANR1I2NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265406-B1 VIRICIDES DUPONT PHARMACEUTICALS COMPANY 2001-07-24 US disclosed
US-6090821-A ENZYME INHIBITORS; VIRICIDES E. I. DUPONT DE NEMOURS AND COMPANY (US) 2000-07-18 US disclosed