SCHEMBL7994083

SCHEMBL7994083

CC1=NN(C)CCN1c1ccc(N2C[C@H](CNC(=O)C3CC=C(Cl)S3)OC2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F10 P00742 19/20 0.45
MAOA P21397 1/20 0.42
F2 P00734 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ABCB11 O95342 1/20 0.42
ST14 Q9Y5Y6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7983045 0.87 F10 (0.44) F10MAOA
SCHEMBL7983038 0.86 F10 (0.48) F10F2CYP1A2CYP3A4CYP2D6
SCHEMBL7995877 0.86 F10 (0.45) F10F2CYP1A2CYP3A4CYP2D6
SCHEMBL7982207 0.85 F10 (0.42) F10
SCHEMBL7997062 0.84 F10 (0.44) F10F2CYP1A2CYP3A4CYP2D6
SCHEMBL7997701 0.83 F10 (0.45) F10MAOAF2ABCB11ST14
SCHEMBL7992863 0.83 F10 (0.44) F10F2CYP1A2CYP3A4CYP2D6
SCHEMBL8000437 0.81 F10 (0.47) F10F2ABCB11ST14
SCHEMBL4761202 0.81 F10 (0.70) F10F2ABCB11ST14
SCHEMBL13479673 0.80 F10 (0.66) F10MAOAABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010002115-A2 FXA INHIBITORS WITH CYCLIC AMIDOXIME OR CYCLIC AMIDRAZONE AS P4 SUBUNIT, PROCESSES FOR THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS AND DERIVATIVES THEREOF LEGOCHEM BIOSCIENCE LTD. (KR) 2010-01-07 WO disclosed