SCHEMBL7995271

SCHEMBL7995271

C/C=C(/Oc1c(F)cc(Cl)cc1F)c1nnc(-c2ccc3c(c2)CN(Cc2ccc(OC)cc2)C3=O)n1C1CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 2/20 0.35
TOP2A P11388 1/20 0.32
TOP2B Q02880 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE1C Q14123 1/20 0.32
TP53 P04637 1/20 0.32
MAOA P21397 2/20 0.32
MAPK1 P28482 2/20 0.32
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
FAAH O00519 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
ABHD6 Q9BV23 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968696 0.81 TNIK (0.35) TNIKTP53MAPK1GRM2
SCHEMBL7985372 0.75 TNIK (0.35) TNIKGRM2
SCHEMBL7981460 0.74 TNIK (0.37) TNIKPSEN1PSEN2APH1BNCSTN
SCHEMBL7968271 0.74 TP53 (0.35) PDE1APDE1BPDE1CTP53MAPK1
SCHEMBL7968654 0.74 TNIK (0.37) TNIKMAPK1GRM2
SCHEMBL7985423 0.73 TNIK (0.36) TNIKMEN1KMT2A
SCHEMBL7985804 0.68 TP53 (0.37) PDE1APDE1BPDE1CTP53LMNA
SCHEMBL12671374 0.68 CYP19A1 (0.43)
SCHEMBL14991264 0.68 GAA (0.47) TNIKTP53MAPK1LMNAHTT
SCHEMBL7995270 0.67 IDH1 (0.33) LMNAHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001946-A1 TRIAZOLE DERIVATIVE OR SALT THEREOF アステラス製薬株式会社 (JP) 2010-01-07 WO disclosed