SCHEMBL7999219

SCHEMBL7999219

N#Cc1c(Cl)nc2[nH]c(=O)[nH]c(=O)c2c1-c1ccc(CCCO)cc1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 9/20 0.45
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
P2RY12 Q9H244 2/20 0.42
TDO2 P48775 1/20 0.38
NPSR1 Q6W5P4 1/20 0.35
PDE9A O76083 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ACMSD Q8TDX5 1/20 0.33
XDH P47989 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1177330 0.83 IDO1 (0.45) IDO1PDE3BPDE3AP2RY12TDO2
SCHEMBL1177647 0.81 IDO1 (0.59) IDO1TDO2PDE9AALDH1A1
SCHEMBL1176947 0.73 KDM4E (0.45) IDO1PDE3BPDE3AP2RY12NPSR1
SCHEMBL8009392 0.71 PDE3B (0.45) IDO1PDE3BPDE3AP2RY12
SCHEMBL1176944 0.69 IDO1 (0.59) IDO1TDO2ALDH1A1XDH
SCHEMBL12163763 0.66 ADORA1 (0.51) NPSR1ALDH1A1
SCHEMBL12163643 0.65 ADORA1 (0.47) NPSR1ALDH1A1
SCHEMBL8032685 0.64 ADORA1 (0.49) ACMSD
SCHEMBL10194179 0.64 ADORA1 (0.64) ACMSD
SCHEMBL14498361 0.63 IDO1 (0.51) IDO1NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080198-A1 FUSED CYNOPRYRIDINES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed