SCHEMBL8003035

SCHEMBL8003035

N#Cc1c(NC[C@H](O)CO)nc(SCc2csc(-c3ccc(Cl)cc3)n2)c(C#N)c1-c1nccs1

nearest known ligand 0.53

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 19/20 0.53
SLC6A3 Q01959 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410928 0.92 ADORA1 (0.57) ADORA1SLC6A3
SCHEMBL1074200 0.86 ADORA1 (0.55) ADORA1SLC6A3
SCHEMBL8002794 0.85 ADORA1 (0.53) ADORA1SLC6A3
SCHEMBL12376555 0.84 ADORA1 (0.49) ADORA1SLC6A3
SCHEMBL7999946 0.83 ADORA1 (0.49) ADORA1SLC6A3
SCHEMBL7999947 0.83 ADORA1 (0.61) ADORA1SLC6A3
SCHEMBL8006123 0.82 ADORA1 (0.73) ADORA1SLC6A3
SCHEMBL12376548 0.80 ADORA1 (0.49) ADORA1SLC6A3
SCHEMBL2281758 0.79 ADORA1 (0.63) ADORA1SLC6A3
SCHEMBL12376497 0.78 ADORA1 (0.56) ADORA1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274299-B1 HETEROARYL-SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF FOR TREATMENT OF CARDIOVASCULAR DISEASES BAYER IP GMBH (DE) 2016-06-15 EP disclosed
WO-2009112155-A1 HETEROARYL-SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF FOR TREATMENT OF CARDIOVASCULAR DISEASES BAYER SCHERING PHARMA AG (DE) 2009-09-17 WO disclosed