SCHEMBL8006099

SCHEMBL8006099

N#Cc1c(SCc2csc(-c3ccc(Cl)cc3)n2)nc(N2CC(O)C2)c(C#N)c1-c1cc[nH]n1

nearest known ligand 0.53

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 20/20 0.53
SLC6A3 Q01959 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410903 0.92 ADORA1 (0.53) ADORA1SLC6A3
SCHEMBL1076310 0.85 ADORA1 (0.61) ADORA1SLC6A3
SCHEMBL2282177 0.84 ADORA1 (0.73) ADORA1SLC6A3
SCHEMBL8002243 0.84 ADORA1 (0.55) ADORA1SLC6A3
SCHEMBL1076183 0.84 ADORA1 (0.57) ADORA1SLC6A3
SCHEMBL8001636 0.84 ADORA1 (0.51) ADORA1SLC6A3
SCHEMBL8005108 0.83 ADORA1 (0.52) ADORA1SLC6A3
SCHEMBL924730 0.82 ADORA1 (0.56) ADORA1SLC6A3
SCHEMBL924731 0.82 ADORA1 (0.56) ADORA1SLC6A3
SCHEMBL2277947 0.81 ADORA1 (0.59) ADORA1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274299-B1 HETEROARYL-SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF FOR TREATMENT OF CARDIOVASCULAR DISEASES BAYER IP GMBH (DE) 2016-06-15 EP disclosed
US-8426602-B2 Heteroaryl-substituted dicyanopyridines and their use BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-04-23 US disclosed
WO-2009112155-A1 HETEROARYL-SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF FOR TREATMENT OF CARDIOVASCULAR DISEASES BAYER SCHERING PHARMA AG (DE) 2009-09-17 WO disclosed