SCHEMBL8006696

SCHEMBL8006696

CN1C=C(/C=C/CCN)C=C(OCc2ccccc2)C1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.35
HRH4 Q9H3N8 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
TP53 P04637 1/20 0.34
CHRNA7 P36544 2/20 0.34
MAPT P10636 1/20 0.34
KDM1A O60341 4/20 0.33
MAOB P27338 1/20 0.32
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3712772 0.82
SCHEMBL5196585 0.79
SCHEMBL8016760 0.76
SCHEMBL23070558 0.67 HTT (0.40) HTTHRH4NPC1RAB9AHRH3
SCHEMBL1536706 0.58 IDO1 (0.54) MAOBIDO1
SCHEMBL5682418 0.58 IDO1 (0.54) MAOBIDO1
SCHEMBL1829198 0.58 IDO1 (0.54) MAOBIDO1
SCHEMBL8553314 0.57 HTR2A (0.58) MAOB
SCHEMBL5956337 0.57 MAOB (0.68) MAOBIDO1
SCHEMBL8556069 0.57 HTR2A (0.58) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973743-A1 PHARMACEUTICAL COMPOSITIONS INCORPORATING ARYL SUBSTITUTED OLEFINIC AMINE COMPOUNDS R.J. REYNOLDS TOBACCO COMPANY (US) 2000-01-26 EP claimed
WO-1998037071-A1 PHARMACEUTICAL COMPOSITIONS INCORPORATING ARYL SUBSTITUTED OLEFINIC AMINE COMPOUNDS R.J. REYNOLDS TOBACCO COMPANY (US) 1998-08-27 WO claimed