SCHEMBL8009055

SCHEMBL8009055

CCc1nc2c(cnn2CC)c(NC2CCOCC2)c1CNC(=O)NCc1ccc(Cl)c(-c2cccc(CN3CCN[C@H](C)C3)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 18/20 0.46
PDE4B Q07343 1/20 0.42
CHRM2 P08172 6/20 0.42
CHRM1 P11229 6/20 0.42
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4361960 0.97 CHRM3 (0.46) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL4362581 0.97 CHRM3 (0.46) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL13750945 0.96 CHRM3 (0.44) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL4353957 0.96 CHRM3 (0.45) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL4350682 0.96 CHRM3 (0.45) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL4099043 0.94 CHRM3 (0.47) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL1364144 0.94 CHRM3 (0.52) CHRM3CHRM2CHRM1KCNH2
SCHEMBL4093724 0.94 CHRM3 (0.47) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL3426553 0.94 CHRM3 (0.46) CHRM3PDE4BCHRM2CHRM1KCNH2
SCHEMBL8010849 0.94 PDE4B (0.43) CHRM3PDE4BCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100170-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed