SCHEMBL8009592

SCHEMBL8009592

CCc1nc(-c2ccc(N/C(=C3\C(=O)Nc4ccc([N+](=O)[O-])cc43)c3ccc(CCNC(C)=O)cc3)cc2)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.36
KMT2A Q03164 4/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
AKT2 P31751 3/20 0.35
PDPK1 O15530 1/20 0.35
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
EGFR P00533 1/20 0.35
CNR1 P21554 1/20 0.34
MEN1 O00255 3/20 0.33
MAPT P10636 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GSK3B P49841 1/20 0.33
PIN1 Q13526 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009597 1.00 NQO2 (0.36) NQO2KMT2ANPC1RAB9AAKT2
SCHEMBL8016476 0.96 KMT2A (0.35) NQO2KMT2ANPC1RAB9AAKT2
SCHEMBL8016472 0.96 KMT2A (0.35) NQO2KMT2ANPC1RAB9AAKT2
SCHEMBL8001456 0.93 AKT2 (0.41) AKT2PDPK1CA12CA1CA2
SCHEMBL8001454 0.93 AKT2 (0.41) AKT2PDPK1CA12CA1CA2
SCHEMBL8009531 0.92 NQO2 (0.38) NQO2KMT2ANPC1RAB9AAKT2
SCHEMBL8009527 0.92 NQO2 (0.38) NQO2KMT2ANPC1RAB9AAKT2
SCHEMBL8001154 0.90 EGFR (0.37) KMT2AAKT2PDPK1CA12CA1
SCHEMBL8001158 0.90 EGFR (0.37) KMT2AAKT2PDPK1CA12CA1
SCHEMBL8012465 0.89 CA12 (0.36) KMT2AAKT2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO disclosed