SCHEMBL8010335

SCHEMBL8010335

O=[N+]([O-])C=Cc1cc(OCc2ccccc2)c(OCc2ccccc2)cc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 5/20 0.54
TLR2 O60603 5/20 0.54
MAOA P21397 5/20 0.54
MAOB P27338 5/20 0.54
MAPT P10636 6/20 0.54
HPGD P15428 3/20 0.54
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
LMNA P02545 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
NPSR1 Q6W5P4 3/20 0.54
HTT P42858 2/20 0.54
BACE1 P56817 1/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
ALDH1A1 P00352 4/20 0.46
POLB P06746 2/20 0.45
CTSV O60911 1/20 0.44
CTSL P07711 1/20 0.44
HSP90AA1 P07900 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8010330 1.00 TLR4 (0.54) TLR4TLR2MAOAMAOBMAPT
SCHEMBL15952706 0.94 MAPT (0.53) TLR4TLR2MAOAMAOBMAPT
SCHEMBL187779 0.94 MAPT (0.53) TLR4TLR2MAOAMAOBMAPT
SCHEMBL187778 0.94 MAPT (0.53) TLR4TLR2MAOAMAOBMAPT
SCHEMBL15952707 0.94 MAPT (0.53) TLR4TLR2MAOAMAOBMAPT
SCHEMBL10542664 0.91 TLR4 (0.47) TLR4TLR2MAOAMAOBMAPT
SCHEMBL10542672 0.91 TLR4 (0.47) TLR4TLR2MAOAMAOBMAPT
SCHEMBL15952366 0.90 MAPT (0.46) TLR4TLR2MAOAMAOBMAPT
SCHEMBL15952365 0.90 MAPT (0.46) TLR4TLR2MAOAMAOBMAPT
SCHEMBL15952467 0.89 MAPT (0.45) TLR4TLR2MAOAMAOBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6160127-A Process for the preparation of substituted indoles BRISTOL-MYERS SQUIBB COMPANY (US) 2000-12-12 US disclosed
EP-0972763-A1 Process for the preparation of substituted indoles Bristol-Myers Squibb Company (US) 2000-01-19 EP disclosed
US-5536865-A Process for the preparation of 5,6-dihydroxyindole and intermediate compounds L'OREAL (FR) 1996-07-16 US disclosed
US-5508464-A NITRATING OF A 4,5-DIBENZYLOXYPHENYLACETONITRILE, FOLLOWED BY DEBENZYLATION, HYDROGENATION AND CYCLIZATION L'OREAL (FR) 1996-04-16 US disclosed
US-5498746-A Process for the preparation of 5,6-dihydroxyindole and intermediate compounds L'OREAL (FR) 1996-03-12 US disclosed
US-5410067-A Catalytic hydrogenation; cyclization L'OREAL (FR) 1995-04-25 US disclosed
US-4595765-A Process for preparing 5,6-dihydroxyindole CLAIROL INCORPORATED (US) 1986-06-17 US disclosed
US-4595765-A Process for preparing 5,6-dihydroxyindole CLAIROL INCORPORATED (US) 1986-06-17 US disclosed