SCHEMBL8012853

SCHEMBL8012853

CCc1nc(-c2ccc(N/C(=C3\C(=O)Nc4ccc([N+](=O)[O-])cc43)c3ccc(CN)cc3)cc2)c[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
AKT2 P31751 3/20 0.37
ALDH1A1 P00352 3/20 0.35
MAPT P10636 3/20 0.35
MPI P34949 2/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
BLM P54132 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CAPN9 O14815 1/20 0.34
CASP3 P42574 1/20 0.34
GSK3B P49841 4/20 0.34
PKM P14618 1/20 0.34
GALK1 P51570 1/20 0.34
SAE1 Q9UBE0 1/20 0.34
UBA2 Q9UBT2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8012859 1.00 EGFR (0.38) EGFRCA12CA1CA2CA9
SCHEMBL8001154 0.94 EGFR (0.37) EGFRCA12CA1CA2CA9
SCHEMBL8001158 0.94 EGFR (0.37) EGFRCA12CA1CA2CA9
SCHEMBL8012465 0.93 CA12 (0.36) EGFRCA12CA1CA2CA9
SCHEMBL8012469 0.93 CA12 (0.36) EGFRCA12CA1CA2CA9
SCHEMBL8016363 0.92 EGFR (0.39) EGFRCA12CA1CA2CA9
SCHEMBL8016360 0.92 EGFR (0.39) EGFRCA12CA1CA2CA9
SCHEMBL8001474 0.91 EGFR (0.40) EGFRCA12CA1CA2CA9
SCHEMBL8001471 0.91 EGFR (0.40) EGFRCA12CA1CA2CA9
SCHEMBL8001456 0.90 AKT2 (0.41) EGFRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed