SCHEMBL8018932

SCHEMBL8018932

CO[C@@H]1CCC2CSC(NC(=O)OC(C)(C)C)=N[C@@]2(c2cc(N)ccc2F)C1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.37
BACE2 Q9Y5Z0 6/20 0.37
KCNH2 Q12809 3/20 0.35
CTSD P07339 2/20 0.35
CYP2D6 P10635 1/20 0.35
BRAF P15056 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2620032 1.00 BACE1 (0.37) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2620038 1.00 BACE1 (0.37) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL8018929 1.00 BACE1 (0.37) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL10288718 1.00 BACE1 (0.37) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2620039 1.00 BACE1 (0.37) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2632314 1.00 BACE1 (0.37) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2619842 0.96 BACE1 (0.36) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL8028459 0.96 BACE1 (0.36) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL8031653 0.96 BACE1 (0.36) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2619843 0.96 BACE1 (0.36) BACE1BACE2KCNH2CTSDCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009091016-A1 CONDENSED AMINODIHYDROTHIAZINE DERIVATIVE EISAI R & D MANAGEMENT CO., LTD. (JP) 2009-07-23 WO disclosed