SCHEMBL8019299

SCHEMBL8019299

CC(C)N=C=NC(C)C.CCN=C=NC(C)N(C)C

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443991 0.94 CYP1A2 (0.39) CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL8537869 0.91 CYP1A2 (0.38) CYP1A2CYP2D6
SCHEMBL7484113 0.84
Hydrochloric Acid SCHEMBL4275672 0.82
SCHEMBL9074979 0.82 CYP1A2 (0.38) CYP1A2CYP2D6
SCHEMBL3626821 0.77 CYP1A2 (0.32) CYP1A2CYP2D6
Dimethylamine SCHEMBL8019309 0.76 CYP1A2 (0.34) CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL1671539 0.75 CYP1A2 (0.31) CYP1A2CYP2D6
SCHEMBL8019304 0.75 CYP1A2 (0.58) CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL6017809 0.72 CYP1A2 (0.32) CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143895-A TETRAHYDROQUINOLINONE COMPOUND TREGA BIOSCIENCES, INC. (US) 2000-11-07 US disclosed
EP-0983507-A1 TRICYCLIC TETRAHYDROQUINOLINE DERIVATIVES AND TRICYCLIC TETRAHYDROQUINOLINE COMBINATORIAL LIBRARIES Trega Biosciences, Inc. (US) 2000-03-08 EP disclosed
US-5925527-A SCREENING NEW PHARMACEUTICALS TREGA BIOSCIENCES, INC. (US) 1999-07-20 US disclosed
WO-1998034111-A1 TRICYCLIC TETRAHYDROQUINOLINE DERIVATIVES AND TRICYCLIC TETRAHYDROQUINOLINE COMBINATORIAL LIBRARIES TREGA BIOSCIENCES, INC. (US) 1998-08-06 WO disclosed