SCHEMBL8019406

SCHEMBL8019406

Cc1ccc(-c2oc3ccc(Cl)cc3c(=O)c2O)cc1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.85
CSNK2A2 P19784 5/20 0.85
CSNK2B P67870 5/20 0.85
CSNK2A1 P68400 5/20 0.85
TP53 P04637 5/20 0.85
MKNK2 Q9HBH9 1/20 0.71
KDM4E B2RXH2 4/20 0.67
HTT P42858 2/20 0.66
LMNA P02545 1/20 0.66
RET P07949 1/20 0.66
TSHR P16473 1/20 0.66
ALOX12 P18054 1/20 0.66
KDR P35968 1/20 0.66
ADORA3 P0DMS8 3/20 0.62
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
CYP3A4 P08684 2/20 0.61
CYP2C9 P11712 1/20 0.61
HSD17B10 Q99714 1/20 0.61
RXFP1 Q9HBX9 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12941005 0.86 MKNK2 (0.75) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL12941170 0.85 CSNK2A2 (0.75) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL7652737 0.83 MEN1 (0.68) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL25239822 0.81 TP53 (0.67) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL8006203 0.81 MAPT (0.57) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL30667420 0.81 MAPT (0.76) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL8709977 0.81 MAPT (0.71) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL4650064 0.80 MAPT (1.00) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL10037935 0.80 TP53 (1.00) MAPTCSNK2A2CSNK2BCSNK2A1TP53
SCHEMBL4648920 0.78 CSNK2A2 (1.00) MAPTCSNK2A2CSNK2BCSNK2A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0666265-B1 PHOSPHONIC DIESTER DERIVATIVE OTSUKA PHARMA CO LTD (JP) 2000-01-26 EP disclosed
US-5527786-A ANTIDIABETIC AGENTS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1996-06-18 US disclosed
EP-0666265-A1 PHOSPHONIC DIESTER DERIVATIVE OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1995-08-09 EP disclosed