SCHEMBL8019796

SCHEMBL8019796

C[C@@]12CCC[C@H]1[C@@H]1CC[C@H]3NC(=O)C(C(=O)NO)C[C@]3(C)[C@H]1CC2

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.43
GRIN2B Q13224 4/20 0.43
NR1I3 Q14994 1/20 0.40
MBOAT4 Q96T53 1/20 0.39
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
SRD5A2 P31213 2/20 0.37
AR P10275 1/20 0.37
SRD5A1 P18405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9647695 0.89 SRD5A2 (0.46) GRIN1GRIN2BNR1I3CDK5CDK5R1
SCHEMBL7609110 0.88 GRIN1 (0.45) GRIN1GRIN2BNR1I3MBOAT4CDK5
SCHEMBL9547062 0.88 GRIN1 (0.45) GRIN1GRIN2BNR1I3MBOAT4CDK5
SCHEMBL9185884 0.87 CDK5 (0.42) GRIN1GRIN2BNR1I3MBOAT4CDK5
SCHEMBL4731758 0.85 SRD5A2 (0.50) GRIN1GRIN2BNR1I3CDK5CDK5R1
SCHEMBL8764684 0.85 GRIN1 (0.38) GRIN1GRIN2BNR1I3
SCHEMBL10699453 0.84 GRIN1 (0.38) GRIN1GRIN2BNR1I3MBOAT4CDK5
SCHEMBL16235951 0.82 NR1I3 (0.41) GRIN1GRIN2BNR1I3CDK5CDK5R1
SCHEMBL9110720 0.82 NR1I3 (0.48) GRIN1GRIN2BNR1I3MBOAT4CDK5
SCHEMBL15549709 0.82 NR1I3 (0.48) GRIN1GRIN2BNR1I3MBOAT4CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970105-A1 PROCESS FOR PREPARING CARBOXAMIDO-4-AZASTEROIDS PHARMACIA & UPJOHN S.p.A. (IT) 2000-01-12 EP disclosed
WO-1999035161-A1 PROCESS FOR PREPARING CARBOXAMIDO-4-AZASTEROIDS PHARMACIA & UPJOHN SPA (IT) 1999-07-15 WO disclosed