SCHEMBL8022698

SCHEMBL8022698

CSc1ccc(-c2ccc(C[C@@H](C#N)NC(=O)[C@@H]3CCCCN3)cc2)cc1N

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.78
CTSK P43235 5/20 0.78
KCNH2 Q12809 3/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041853 0.93 CTSC (0.81) CTSCCTSKKCNH2
SCHEMBL2073440 0.90 CTSC (0.87) CTSCCTSKKCNH2
SCHEMBL1499178 0.90 CTSC (0.87) CTSCCTSKKCNH2
SCHEMBL2072220 0.88 CTSC (1.00) CTSCCTSKKCNH2
SCHEMBL1499191 0.88 CTSC (1.00) CTSCCTSKKCNH2
SCHEMBL8037900 0.85 CTSC (0.68) CTSCCTSKKCNH2
SCHEMBL8039616 0.85 CTSC (0.82) CTSCCTSKKCNH2
SCHEMBL1499010 0.85 CTSC (0.76) CTSCCTSKKCNH2
SCHEMBL8045417 0.85 CTSC (0.72) CTSCCTSKKCNH2
SCHEMBL8037322 0.83 CTSC (0.68) CTSCCTSKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed