SCHEMBL8022906

SCHEMBL8022906

Oc1ccc(CBr)c(Cl)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.48
MAPK1 P28482 1/20 0.48
HIF1A Q16665 3/20 0.37
HPGD P15428 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HSP90AA1 P07900 2/20 0.37
MAPT P10636 2/20 0.37
ALOX15 P16050 2/20 0.37
SLC22A1 O15245 1/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
HSPD1 P10809 1/20 0.37
HSPA5 P11021 1/20 0.37
IDO1 P14902 1/20 0.37
ALOX12 P18054 1/20 0.37
CASP1 P29466 1/20 0.37
HTT P42858 1/20 0.37
BLM P54132 1/20 0.37
HSPE1 P61604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28472354 0.80 CYP3A4 (0.52) CYP3A4MAPK1HIF1AHPGDMEN1
SCHEMBL843869 0.79 TSHR (0.50) CYP3A4MAPK1HIF1AHPGDALOX15
SCHEMBL7743436 0.76 CYP3A4 (0.75) CYP3A4MAPK1HIF1AHPGDMEN1
SCHEMBL31392414 0.76 CYP3A4 (0.75) CYP3A4MAPK1HIF1AHPGDMEN1
SCHEMBL68064 0.76 CYP3A4 (0.75) CYP3A4MAPK1HIF1AHPGDMEN1
SCHEMBL6305999 0.75 CYP3A4 (0.40) CYP3A4MAPK1IDO1
SCHEMBL11195988 0.74 CYP3A4 (0.46) CYP3A4MAPK1HIF1AHPGDMEN1
SCHEMBL9114093 0.73 PRKCI (0.47) CYP3A4MAPK1HIF1AHPGDMEN1
SCHEMBL10917220 0.72
SCHEMBL2335198 0.71 NOTUM (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2757093-A1 GUANIDINOBENZOIC ACID COMPOUND Astellas Pharma Inc. (JP) 2014-07-23 EP disclosed
EP-0971904-A1 NOVEL 1-AMINO-3 BENZYL URACILS BASF AKTIENGESELLSCHAFT (DE) 2000-01-19 EP disclosed
WO-1998042682-A1 NOVEL 1-AMINO-3 BENZYL URACILS BASF AKTIENGESELLSCHAFT (DE) 1998-10-01 WO disclosed