SCHEMBL8023743

SCHEMBL8023743

CC(C)(C)c1ccccc1OC(=O)[C@H]1CC[C@H]2[C@@H]3C(=O)C[C@H]4NC(=O)CC[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 5/20 0.46
SRD5A1 P18405 2/20 0.46
AR P10275 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8016224 0.88 SRD5A1 (0.61) SRD5A2SRD5A1AR
SCHEMBL8006689 0.88 SRD5A2 (0.47) SRD5A2SRD5A1AR
SCHEMBL8017035 0.84 SRD5A2 (0.44) SRD5A2SRD5A1AR
SCHEMBL8018455 0.84 SRD5A2 (0.43) SRD5A2SRD5A1AR
SCHEMBL8020704 0.77 SRD5A2 (0.53) SRD5A2SRD5A1AR
SCHEMBL8020700 0.77 SRD5A2 (0.53) SRD5A2SRD5A1AR
SCHEMBL8016924 0.76 SRD5A1 (0.47) SRD5A2SRD5A1
SCHEMBL8016710 0.76 SRD5A2 (0.64) SRD5A2SRD5A1AR
SCHEMBL8006808 0.75 SRD5A1 (0.62) SRD5A2SRD5A1AR
SCHEMBL8023744 0.75 SRD5A2 (0.39) SRD5A2SRD5A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP disclosed
US-5278159-A Steroid enzyme inhibitor MERCK & CO., INC. (US) 1994-01-11 US disclosed