SCHEMBL8026014

SCHEMBL8026014

COC(=O)CCC(=O)N(c1ccc2c(c1)nc(Cc1ccc(C#N)cc1)n2C)C1CCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACSL1 P33121 2/20 0.45
ITK Q08881 15/20 0.44
CHEK2 O96017 2/20 0.44
PRKCG P05129 2/20 0.44
FLT3 P36888 2/20 0.44
CSNK1D P48730 2/20 0.44
RPS6KA3 P51812 2/20 0.44
DYRK1A Q13627 2/20 0.44
AURKB Q96GD4 2/20 0.44
IRAK4 Q9NWZ3 2/20 0.44
AURKA O14965 1/20 0.44
MAP4K4 O95819 1/20 0.44
PHKG2 P15735 1/20 0.44
MARK3 P27448 1/20 0.44
CSNK1A1 P48729 1/20 0.44
CLK2 P49760 1/20 0.44
GSK3B P49841 1/20 0.44
IRAK1 P51617 1/20 0.44
NEK4 P51957 1/20 0.44
CSNK1G2 P78368 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8032235 0.85 F2 (0.52) ACSL1
SCHEMBL8029597 0.85 ACSL1 (0.43) ACSL1ITKCHEK2PRKCGFLT3
SCHEMBL8030145 0.81 ACSL1 (0.41) ACSL1ITKCHEK2PRKCGFLT3
SCHEMBL8026495 0.79 ACSL1 (0.42) ACSL1ITKCHEK2PRKCGFLT3
Hydrochloric Acid SCHEMBL8016636 0.78 F2 (0.57) ACSL1CNR2
SCHEMBL8029894 0.77 ITK (0.43) ACSL1ITKCHEK2PRKCGFLT3
SCHEMBL8016122 0.77 F2 (0.57)
SCHEMBL8027050 0.77 ITK (0.45) ACSL1ITKCHEK2PRKCGFLT3
Hydrochloric Acid SCHEMBL8029528 0.76 F2 (0.56)
SCHEMBL8132612 0.75 ITK (0.38) ACSL1ITKCHEK2PRKCGFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060166-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS Boehringer Ingelheim Pharma KG (DE) 2000-12-20 EP disclosed
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed
WO-1999040072-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-08-12 WO disclosed