SCHEMBL8029083

SCHEMBL8029083

CCCCCCc1ccc2ccc(OCc3ccc4ccccc4n3)cc2c1O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYSLTR1 Q9Y271 11/20 0.61
CYSLTR2 Q9NS75 7/20 0.61
GPBAR1 Q8TDU6 5/20 0.61
MAPK1 P28482 2/20 0.56
CYP1A2 P05177 2/20 0.56
ALOX5 P09917 2/20 0.56
TP53 P04637 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
TSHR P16473 1/20 0.56
NFKB1 P19838 1/20 0.56
CYP2C19 P33261 1/20 0.56
HIF1A Q16665 1/20 0.56
MEN1 O00255 1/20 0.56
GMNN O75496 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
HPGD P15428 1/20 0.56
PTGS1 P23219 1/20 0.56
PTGS2 P35354 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10632839 0.79 GPBAR1 (0.76) CYSLTR1CYSLTR2GPBAR1MAPK1CYP1A2
SCHEMBL15271902 0.78 GPBAR1 (0.77) CYSLTR1CYSLTR2GPBAR1MAPK1CYP1A2
SCHEMBL8029305 0.77 PDE10A (0.52) CYSLTR1CYSLTR2GPBAR1ALOX5PDE10A
Ammonia Solution, Strong SCHEMBL9585183 0.77 CYSLTR1 (0.69) CYSLTR1CYSLTR2GPBAR1MAPK1CYP1A2
SCHEMBL10544630 0.76 CYSLTR1 (0.84) CYSLTR1CYSLTR2GPBAR1MAPK1CYP1A2
SCHEMBL9208722 0.76 CYSLTR1 (0.60) CYSLTR1CYSLTR2GPBAR1MAPK1CYP1A2
SCHEMBL31058301 0.75 TYR (0.47) ALOX5TP53CYP3A4TSHRMEN1
SCHEMBL11825062 0.75 TYR (0.47) ALOX5TP53CYP3A4TSHRMEN1
SCHEMBL25205081 0.75 TYR (0.54) CYP3A4ALDH1A1HPGD
SCHEMBL11134384 0.75 TYR (0.54) CYP3A4ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166031-A Substituted tetralins, chromans and related compounds in the treatment of asthma PFIZER INC, (US) 2000-12-26 US disclosed
WO-1989003681-A1 SUBSTITUTED TETRALINS, CHROMANS AND RELATED COMPOUNDS IN THE TREATMENT OF ASTHMA PFIZER INC. (US) 1989-05-05 WO disclosed