SCHEMBL8029409

SCHEMBL8029409

Cc1cc(=O)oc2cc(OCc3ccccc3)c(O)cc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.72
RAB9A P51151 3/20 0.64
NPC1 O15118 2/20 0.64
CASP3 P42574 2/20 0.64
SENP8 Q96LD8 2/20 0.64
SENP7 Q9BQF6 2/20 0.64
SENP6 Q9GZR1 2/20 0.64
PKM P14618 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.64
MAOA P21397 1/20 0.64
TDP1 Q9NUW8 1/20 0.64
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
MCL1 Q07820 2/20 0.55
CYP3A4 P08684 1/20 0.55
THRB P10828 1/20 0.55
AKR1B1 P15121 1/20 0.55
HPGD P15428 1/20 0.55
HSD17B10 Q99714 1/20 0.55
MAPT P10636 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13561098 0.90 MAOB (0.70) MAOBRAB9ANPC1CASP3SENP8
SCHEMBL7299491 0.81 KDM4E (0.62) NPC1KDM4EALDH1A1MCL1CYP3A4
SCHEMBL6702416 0.79 CA9 (0.64) MAOBNPC1MAOAKDM4EALDH1A1
SCHEMBL31293440 0.79 KDM4E (0.56) MAOBNPC1KDM4EALDH1A1MCL1
SCHEMBL107774 0.78 MAOB (1.00) MAOBRAB9ANPC1CASP3SENP8
SCHEMBL29382160 0.78 MAOB (1.00) MAOBRAB9ANPC1CASP3SENP8
SCHEMBL8807762 0.77 KDM4E (0.70) MAOBMAOAKDM4EALDH1A1MCL1
SCHEMBL11095625 0.76 HSD17B3 (0.63) MAOBRAB9ANPC1CASP3SENP8
Metesculetol SCHEMBL29649664 0.75 KDM4E (0.62) MAOBKDM4EALDH1A1MCL1CYP3A4
Metesculetol SCHEMBL1053452 0.75 KDM4E (0.62) MAOBKDM4EALDH1A1MCL1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1053193-C Esculetin derivatives, process for manufacture and use thereof, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 2000-06-07 CN disclosed
EP-0654479-B1 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 2000-03-15 EP disclosed
CN-1106398-A Esculetin derivatives, process for manufacture and use thereof, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 1995-08-09 CN disclosed
EP-0654479-A2 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-05-24 EP disclosed