SCHEMBL8030588

SCHEMBL8030588

NC1=NC2(c3cc(NC(=O)c4ccc(C(F)(F)F)cn4)ccc3F)CCCC2CS1

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.81
BACE2 Q9Y5Z0 8/20 0.81
KCNH2 Q12809 3/20 0.57
CYP2D6 P10635 1/20 0.57
CTSD P07339 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2620251 1.00 BACE1 (0.81) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL2934242 0.97 BACE1 (0.77) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL2620187 0.97 BACE1 (0.77) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL2620313 0.97 BACE1 (0.76) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL2926576 0.97 BACE1 (0.76) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL8035114 0.97 BACE1 (0.76) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL2925371 0.90 BACE1 (1.00) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL8033554 0.90 BACE1 (0.87) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL2620096 0.90 BACE1 (0.87) BACE1BACE2KCNH2CYP2D6CTSD
SCHEMBL2620100 0.90 BACE1 (1.00) BACE1BACE2KCNH2CYP2D6CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233474-B1 CONDENSED AMINODIHYDROTHIAZINE DERIVATIVE EISAI R&D MAN CO LTD (JP) 2015-08-05 EP disclosed
WO-2009091016-A1 CONDENSED AMINODIHYDROTHIAZINE DERIVATIVE EISAI R & D MANAGEMENT CO., LTD. (JP) 2009-07-23 WO disclosed