SCHEMBL8030658

SCHEMBL8030658

CO[N+](=O)c1ccc(F)c(C23CCCCC2CSC(NC(=O)OC(C)(C)C)=N3)c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.41
BACE2 Q9Y5Z0 7/20 0.41
BRAF P15056 1/20 0.32
CTSD P07339 4/20 0.31
KCNH2 Q12809 2/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2619801 0.92 BACE1 (0.41) BACE1BACE2BRAFCTSDKCNH2
SCHEMBL10288284 0.91 BACE2 (0.41) BACE1BACE2BRAF
SCHEMBL2619815 0.91 BACE2 (0.41) BACE1BACE2BRAF
SCHEMBL2619800 0.91 BACE2 (0.41) BACE1BACE2BRAF
SCHEMBL8018699 0.90 BACE2 (0.41) BACE1BACE2BRAF
SCHEMBL2619816 0.90 BACE2 (0.41) BACE1BACE2BRAF
SCHEMBL2619807 0.89 BACE2 (0.43) BACE1BACE2BRAFKCNH2CYP2D6
SCHEMBL13177589 0.88 BACE1 (0.34) BACE1BACE2BRAFCTSDKCNH2
SCHEMBL8034905 0.87 BACE1 (0.38) BACE1BACE2CTSDKCNH2CYP2D6
SCHEMBL15171566 0.87 BACE1 (0.44) BACE1BACE2BRAFCTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009091016-A1 CONDENSED AMINODIHYDROTHIAZINE DERIVATIVE EISAI R & D MANAGEMENT CO., LTD. (JP) 2009-07-23 WO disclosed