SCHEMBL8033943

SCHEMBL8033943

Clc1cnc(Sc2nnc(-c3cccs3)n2-c2ccccc2)s1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 8/20 0.61
HSD17B10 Q99714 7/20 0.59
KDM4E B2RXH2 4/20 0.59
ALDH1A1 P00352 4/20 0.56
MAPK1 P28482 2/20 0.56
NPSR1 Q6W5P4 6/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
RECQL P46063 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HPGD P15428 2/20 0.47
PPARG P37231 2/20 0.47
RXFP1 Q9HBX9 2/20 0.47
NR2E3 Q9Y5X4 2/20 0.47
NCOR2 Q9Y618 2/20 0.47
HTT P42858 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042736 0.91 TSHR (0.52) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8043144 0.90 TSHR (0.50) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8042619 0.89 TSHR (0.57) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8050287 0.89 HSD17B10 (0.53) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8033911 0.87 TSHR (0.48) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8048248 0.87 NPSR1 (0.51) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8043564 0.87 TSHR (0.48) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8046532 0.86 TSHR (0.48) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8034049 0.84 TSHR (0.58) TSHRHSD17B10KDM4EALDH1A1MAPK1
SCHEMBL8044235 0.83 TSHR (0.43) TSHRHSD17B10KDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed