SCHEMBL8037320

SCHEMBL8037320

C[S+]([O-])c1cc(-c2ccc(C[C@@H](C#N)NC(=O)[C@@H]3CCCCN3C(=O)OC(C)(C)C)cc2)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 19/20 0.43
KCNH2 Q12809 4/20 0.42
CTSK P43235 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2072277 0.91 CTSC (0.49) CTSCKCNH2CTSK
SCHEMBL2072280 0.91 CTSC (0.49) CTSCKCNH2CTSK
SCHEMBL8036268 0.87 CTSC (0.49) CTSCKCNH2CTSK
SCHEMBL8041807 0.87 CTSC (0.52) CTSCKCNH2CTSK
SCHEMBL2072370 0.83 CTSC (0.47) CTSCKCNH2CTSK
SCHEMBL2072367 0.83 CTSC (0.47) CTSCKCNH2CTSK
SCHEMBL8041661 0.83 CTSC (0.43) CTSCKCNH2CTSK
SCHEMBL7858085 0.82 CTSC (0.55) CTSCKCNH2CTSK
SCHEMBL2073293 0.82 CTSC (0.55) CTSCKCNH2CTSK
SCHEMBL2073295 0.82 CTSC (0.55) CTSCKCNH2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed