SCHEMBL8039004

SCHEMBL8039004

CCc1ccc(-c2ccc(C[C@@H](N)NC(=O)[C@@H]3CCCCN3)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSC P53634 11/20 0.58
CTSK P43235 4/20 0.58
KCNH2 Q12809 2/20 0.58
HTR2C P28335 2/20 0.44
HTR2B P41595 1/20 0.41
GHSR Q92847 3/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
DPP7 Q9UHL4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8039150 0.90 CTSC (0.59) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8040349 0.86 CTSC (0.66) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8036119 0.86 CTSC (0.55) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL7857540 0.84 CTSC (0.52) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL8031912 0.84 CTSC (0.56) CTSCCTSKKCNH2HTR2CGHSR
SCHEMBL8039503 0.84 CTSC (0.51) CTSCCTSKKCNH2HTR2CGHSR
SCHEMBL12422428 0.84 CTSC (0.82) CTSCCTSKKCNH2
SCHEMBL8023034 0.83 CTSC (0.52) CTSCCTSKKCNH2HTR2CHTR2B
SCHEMBL12844186 0.83 CTSC (0.57) CTSCCTSKKCNH2HTR2CGHSR
SCHEMBL8034395 0.82 CTSC (0.49) CTSCCTSKKCNH2HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed