SCHEMBL8039617

SCHEMBL8039617

CCCS(=O)(=O)c1ccc(-c2ccc(C[C@@H](C#N)NC(=O)[C@@H]3CCCCN3)cc2)cc1N

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.64
CTSK P43235 5/20 0.64
KCNH2 Q12809 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031971 0.94 CTSC (0.64) CTSCCTSKKCNH2
SCHEMBL12383379 0.90 CTSC (0.68) CTSCCTSKKCNH2
SCHEMBL8037900 0.90 CTSC (0.68) CTSCCTSKKCNH2
SCHEMBL2075351 0.89 CTSC (0.70) CTSCCTSKKCNH2
SCHEMBL1499070 0.89 CTSC (0.70) CTSCCTSKKCNH2
SCHEMBL8036052 0.88 CTSC (0.67) CTSCCTSKKCNH2
SCHEMBL8037322 0.85 CTSC (0.68) CTSCCTSKKCNH2
SCHEMBL3689684 0.83 CTSC (0.75) CTSCCTSKKCNH2
SCHEMBL3689681 0.83 CTSC (0.75) CTSCCTSKKCNH2
SCHEMBL1499099 0.83 CTSC (0.73) CTSCCTSKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed