SCHEMBL8040069

SCHEMBL8040069

N#Cc1cc(CN2CC[C@H](N)C2=O)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
DPP4 P27487 3/20 0.39
DPP8 Q6V1X1 1/20 0.39
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
KCNH2 Q12809 3/20 0.35
CYP3A4 P08684 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34
CHKA P35790 1/20 0.34
KDM1A O60341 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7214287 0.84 CYP3A4 (0.36) CYP3A4
SCHEMBL8040065 0.83 TNKS (0.43) TNKSTNKS2DPP4DPP8KCNH2
SCHEMBL7424938 0.80 FNTA (0.47) DPP4DPP8KCNH2CYP3A4FNTA
Hydrochloric Acid SCHEMBL2328814 0.79 FNTA (0.47) DPP4DPP8KCNH2CYP3A4FNTA
Hydrochloric Acid SCHEMBL2328817 0.79 FNTA (0.47) DPP4DPP8KCNH2CYP3A4FNTA
SCHEMBL7482530 0.78 SIRT2 (0.48) DPP4DPP8KCNH2CYP3A4FNTA
SCHEMBL7423151 0.78 KDM4E (0.35) DPP4DPP8KCNH2CYP3A4FNTA
SCHEMBL7419120 0.78 SIRT2 (0.48) DPP4DPP8KCNH2CYP3A4FNTA
SCHEMBL7424077 0.78 KDM4E (0.35) DPP4DPP8KCNH2CYP3A4FNTA
Hydrochloric Acid SCHEMBL8040100 0.77 KDM4E (0.35) DPP4DPP8KCNH2CYP3A4FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6034093-A Substituted sulfonic acid N-[(aminoiminomethyl)phenylalkyl]-azaheterocyclylamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 2000-03-07 US disclosed