SCHEMBL8041102

SCHEMBL8041102

COc1cc(-c2noc(C)n2)c(C=O)cc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.41
MAPT P10636 8/20 0.40
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 2/20 0.37
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
AOX1 Q06278 1/20 0.37
TRIM24 O15164 1/20 0.37
ALDH5A1 P51649 1/20 0.37
ABAT P80404 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TRIM33 Q9UPN9 1/20 0.37
NPC1 O15118 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
POLB P06746 1/20 0.36
TP53 P04637 1/20 0.36
MAOA P21397 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5883322 0.89 KDM4E (0.46) ERN1MAPTALDH1A1KDM4EHSD17B10
SCHEMBL1618138 0.85 MAPT (0.42) ERN1MAPTALDH1A1KDM4EHSD17B10
SCHEMBL12717346 0.84 MAPT (0.46) MAPTALDH1A1KDM4EHSD17B10HPGD
SCHEMBL8037443 0.82 MAPT (0.40) MAPTALDH1A1KDM4EHSD17B10HPGD
SCHEMBL8044102 0.79 MAPT (0.42) MAPTALDH1A1KDM4EHSD17B10HPGD
SCHEMBL8037487 0.79 MAPT (0.42) MAPTALDH1A1KDM4EHSD17B10HPGD
SCHEMBL1617931 0.78 MAPT (0.41) MAPTALDH1A1KDM4EHSD17B10HPGD
SCHEMBL8037477 0.78 MAPT (0.44) MAPTALDH1A1KDM4EHSD17B10HPGD
SCHEMBL12717344 0.76 S1PR1 (0.46) MAPTALDH1A1KDM4EHSD17B10HPGD
SCHEMBL12717352 0.76 S1PR1 (0.41) MAPTALDH1A1KDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246338-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, USE OF THE CATECHOL DERIVATIVE, AND USE OF THE PHARMACEUTICAL COMPOSITION Kissei Pharmaceutical Co., Ltd. (JP) 2010-11-03 EP disclosed
WO-2009081891-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, USE OF THE CATECHOL DERIVATIVE, AND USE OF THE PHARMACEUTICAL COMPOSITION KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed