SCHEMBL8041706

SCHEMBL8041706

[CH2]c1ccc(OCc2cccnc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.56
CYP19A1 P11511 1/20 0.50
CYP11B1 P15538 1/20 0.50
CYP11B2 P19099 1/20 0.50
GPR132 Q9UNW8 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TP53 P04637 1/20 0.48
POLB P06746 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HTR1A P08908 1/20 0.48
DRD2 P14416 1/20 0.48
RAB9A P51151 1/20 0.47
MMP13 P45452 2/20 0.46
MAOA P21397 2/20 0.46
ACACB O00763 1/20 0.46
KDM1A O60341 1/20 0.46
F9 P00740 1/20 0.46
F10 P00742 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28048524 0.91 MAPK1 (0.64) MAPK1CYP19A1CYP11B1CYP11B2GPR132
SCHEMBL7311175 0.84 MAPK1 (0.65) MAPK1GPR132MEN1KMT2AHTR1A
SCHEMBL8881389 0.83 HTT (0.62) MAPK1CYP19A1CYP11B1CYP11B2GPR132
SCHEMBL171895 0.83 MAPK1 (0.56) MAPK1CYP19A1CYP11B1CYP11B2GPR132
SCHEMBL18297474 0.83 APP (0.58) MAPK1CYP19A1CYP11B1CYP11B2GPR132
SCHEMBL30354931 0.83 MAOB (0.62) MAPK1CYP19A1CYP11B1CYP11B2GPR132
SCHEMBL3761776 0.83 MAOB (0.62) MAPK1CYP19A1CYP11B1CYP11B2GPR132
SCHEMBL8361615 0.83 MAPK1 (0.56) MAPK1CYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL4060132 0.83 MAPK1 (0.56) MAPK1CYP19A1CYP11B1CYP11B2GPR132
SCHEMBL5392025 0.81 MAPK1 (0.58) MAPK1CYP19A1CYP11B1CYP11B2GPR132

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0707564-B1 DIFLUORO STATONE ANALOGS MERRELL PHARMA INC (US) 2000-09-20 EP claimed
US-5948778-A Difluoro statone antiviral analogs MERREL PHARMACEUTICALS INC. (US) 1999-09-07 US claimed