SCHEMBL8041745

SCHEMBL8041745

CC(C1CCN(C(=O)c2ncc(C(F)(F)F)cc2S(C)(=O)=O)CC1)S(=O)(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 20/20 0.62
NR1I2 O75469 10/20 0.51
CYP3A4 P08684 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3038851 1.00 CACNA1B (0.62) CACNA1BNR1I2CYP3A4
SCHEMBL13221164 1.00 CACNA1B (0.62) CACNA1BNR1I2CYP3A4
SCHEMBL13221172 0.91 CACNA1B (0.56) CACNA1BNR1I2CYP3A4
SCHEMBL3039554 0.91 CACNA1B (0.56) CACNA1BNR1I2CYP3A4
SCHEMBL3030001 0.89 CACNA1B (0.58) CACNA1BNR1I2CYP3A4
SCHEMBL8044416 0.89 CACNA1B (0.58) CACNA1BNR1I2CYP3A4
SCHEMBL3045391 0.85 CACNA1B (0.73) CACNA1BNR1I2CYP3A4
SCHEMBL3035131 0.85 CACNA1B (0.67) CACNA1BNR1I2CYP3A4
SCHEMBL3025680 0.81 CACNA1B (0.73) CACNA1BNR1I2CYP3A4
SCHEMBL12542551 0.81 CACNA1B (0.44) CACNA1BNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009045382-A1 SUBSTITUTED ARYL SULFONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2009-04-09 WO disclosed