SCHEMBL8043616

SCHEMBL8043616

CCCc1c(F)cccc1C1CCN(c2ccn3c(CC(F)(F)F)cnc3c2C#N)CC1

nearest known ligand 0.66

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 20/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL924110 0.86 GRM2 (0.70) GRM2
SCHEMBL921945 0.86 GRM2 (0.75) GRM2
SCHEMBL8053278 0.82 GRM2 (0.74) GRM2
SCHEMBL924146 0.81 GRM2 (0.71) GRM2
SCHEMBL8045719 0.80 GRM2 (0.57) GRM2
SCHEMBL921967 0.80 GRM2 (1.00) GRM2
SCHEMBL3652536 0.79 GRM2 (0.68) GRM2
SCHEMBL922899 0.74 GRM2 (1.00) GRM2
SCHEMBL12907972 0.72 GRM2 (0.58) GRM2
SCHEMBL748766 0.72 GRM2 (0.81) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009062676-A2 IMIDAZO[1,2-A]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC. (US) 2009-05-22 WO disclosed