SCHEMBL8043701

SCHEMBL8043701

Sc1nnc(-c2cncc(Br)c2)s1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.42
PTK2 Q05397 1/20 0.41
HDAC6 Q9UBN7 1/20 0.38
CYP11B2 P19099 3/20 0.34
CYP11B1 P15538 2/20 0.34
POLB P06746 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045495 0.75 HDAC1 (0.46) KDM4ESMN1; SMN2
SCHEMBL10365074 0.75 KDM4E (0.35) CYP2A6KDM4ESMN1; SMN2
SCHEMBL14557095 0.74 SNCA (0.37) KDM4ESMN1; SMN2
SCHEMBL8047389 0.73 CA1 (0.49) KDM4ESMN1; SMN2
SCHEMBL14392676 0.71 CYP2A6 (0.61) CYP2A6PTK2HDAC6CYP11B2CYP11B1
SCHEMBL14557099 0.69 KDM4E (0.43) POLBKDM4ESMN1; SMN2
SCHEMBL31417903 0.69 CYP2A6 (0.44) CYP2A6PTK2HDAC6CYP11B2CYP11B1
SCHEMBL30396089 0.69 KDM4E (0.64) CYP2A6KDM4ESMN1; SMN2
SCHEMBL969939 0.67 KDM4E (0.59) POLBKDM4ESMN1; SMN2
SCHEMBL969945 0.66 PIK3CA (0.40) KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed