SCHEMBL8045547

SCHEMBL8045547

C[C@@H]1CCC[C@@]2(C)CC[C@H]3[C@H](CS)CC[C@@H](C[C@H]12)C3(C)C

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1I3 Q14994 1/20 0.37
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
RET P07949 1/20 0.34
MAPK14 Q16539 1/20 0.34
CAMK1D Q8IU85 1/20 0.34
GRIN1 Q05586 3/20 0.31
GRIN2B Q13224 3/20 0.31
AKR1B10 O60218 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6937047 0.87 CDK5 (0.38) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL27471621 0.87 CDK5 (0.35) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL27933815 0.86 CDK5 (0.35) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL586768 0.86 RET (0.39) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL28286229 0.86 CDK5 (0.35) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL28013347 0.84 CDK5 (0.33) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL5149381 0.84 RET (0.35) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL3825 0.84 CDK5 (0.40) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL332530 0.84 CDK5 (0.40) NR1I3CDK5CDK5R1RETMAPK14
SCHEMBL901326 0.84 CDK5 (0.40) NR1I3CDK5CDK5R1RETMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017935-A 7-sulfur substituted paclitaxels BRISTOL-MYERS SQUIBB COMPANY (US) 2000-01-25 US disclosed
WO-1998047360-A1 7-SULFUR SUBSTITUTED PACLITAXELS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-10-29 WO disclosed